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7LG7

Crystal structure of CoV-2 Nsp3 Macrodomain complex with PARG345

Summary for 7LG7
Entry DOI10.2210/pdb7lg7/pdb
Related7KFP 7KG0 7KG1 7KG3 7KG6 7KG7 7KG8 7KXB
DescriptorNon-structural protein 3, 3-[(1,3-dimethyl-2,6-dioxo-2,3,6,9-tetrahydro-1H-purin-8-yl)sulfanyl]-N-{[2-(morpholin-4-yl)ethyl]sulfonyl}propanamide, SULFATE ION, ... (4 entities in total)
Functional Keywordshydrolase, sars-cov-2, macrodomain
Biological sourceSevere acute respiratory syndrome coronavirus 2 (2019-nCoV, SARS-CoV-2)
Total number of polymer chains1
Total formula weight18959.44
Authors
Arvai, A.,Brosey, C.A.,Bommagani, S.,Link, T.,Jones, D.E.,Ahmed, Z.,Tainer, J.A. (deposition date: 2021-01-19, release date: 2021-02-17, Last modification date: 2023-10-18)
Primary citationBrosey, C.A.,Houl, J.H.,Katsonis, P.,Balapiti-Modarage, L.P.F.,Bommagani, S.,Arvai, A.,Moiani, D.,Bacolla, A.,Link, T.,Warden, L.S.,Lichtarge, O.,Jones, D.E.,Ahmed, Z.,Tainer, J.A.
Targeting SARS-CoV-2 Nsp3 macrodomain structure with insights from human poly(ADP-ribose) glycohydrolase (PARG) structures with inhibitors.
Prog.Biophys.Mol.Biol., 163:171-186, 2021
Cited by
PubMed: 33636189
DOI: 10.1016/j.pbiomolbio.2021.02.002
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

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