7FGT
Discovery of DS15060524; Gene targeting chimera (GeneTAC) for the treatment of Friedreich's Ataxia (FRDA)
Summary for 7FGT
Entry DOI | 10.2210/pdb7fgt/pdb |
Related PRD ID | PRD_002367 |
Descriptor | DNA (5'-D(*AP*AP*GP*AP*AP*GP*AP*AP*G)-3'), DNA (5'-D(*CP*TP*TP*CP*TP*TP*CP*TP*T)-3'), ~{N}-[3-[3-(dimethylamino)propylamino]-3-oxidanylidene-propyl]-1-methyl-4-[3-[[1-methyl-4-[[1-methyl-4-[3-[[1-methyl-4-[(1-methylimidazol-2-yl)carbonylamino]pyrrol-2-yl]carbonylamino]propanoylamino]imidazol-2-yl]carbonylamino]pyrrol-2-yl]carbonylamino]propanoylamino]imidazole-2-carboxamide (3 entities in total) |
Functional Keywords | friedreich's ataxia pip, dna |
Biological source | Homo sapiens More |
Total number of polymer chains | 2 |
Total formula weight | 6383.63 |
Authors | Takase, N.,Kawai, G.,Igarashi, W.,Katagiri, T. (deposition date: 2021-07-28, release date: 2022-08-03, Last modification date: 2024-05-15) |
Primary citation | Igarashi, W.,Takase, N.,Kawai, G.,Katagiri, T. Discovery of DS15060524; Gene targeting chimera (GeneTAC) for the treatment of Friedreich's Ataxia (FRDA) To be published, |
Experimental method | SOLUTION NMR |
Structure validation
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