7F2X
Crystal structure of MEK1 C121S mutant
Summary for 7F2X
Entry DOI | 10.2210/pdb7f2x/pdb |
Descriptor | MEK1 F11, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER (3 entities in total) |
Functional Keywords | kinase, signaling protein |
Biological source | Homo sapiens |
Total number of polymer chains | 1 |
Total formula weight | 36219.26 |
Authors | Fujioka, Y.,Noda, N.N. (deposition date: 2021-06-15, release date: 2022-06-22, Last modification date: 2023-11-29) |
Primary citation | Kubota, Y.,Fujioka, Y.,Patil, A.,Takagi, Y.,Matsubara, D.,Iijima, M.,Momose, I.,Naka, R.,Nakai, K.,Noda, N.N.,Takekawa, M. Qualitative differences in disease-associated MEK mutants reveal molecular signatures and aberrant signaling-crosstalk in cancer. Nat Commun, 13:4063-4063, 2022 Cited by PubMed: 35831322DOI: 10.1038/s41467-022-31690-w PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.007 Å) |
Structure validation
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