7EIK
RD4-BD1 in complex with LT-872-297
Summary for 7EIK
Entry DOI | 10.2210/pdb7eik/pdb |
Descriptor | Bromodomain-containing protein 4, 1-[2-methyl-5-[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-4-(1-methylpyrazol-4-yl)-1H-pyrrol-3-yl]ethanone (3 entities in total) |
Functional Keywords | inhibitor, brd4, bd1, gene regulation |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 15300.69 |
Authors | |
Primary citation | Zheng, W.,Kong, B.,Tang, W.,Zhu, J.,Chen, Y. RD4-BD1 in complex with LT-872-297 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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