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7DYQ

Crystal structure of histone lysine demethylase 4D (KDM4D) in complex with the inhibitor 5-hydroxy-2-methylpyrazolo[1,5-a]pyrido[3,2-e]pyrimidine-3-carbonitrile

Summary for 7DYQ
Entry DOI10.2210/pdb7dyq/pdb
DescriptorLysine-specific demethylase 4D, 5-hydroxy-2-methylpyrazolo[1,5-a]pyrido[3,2-e]pyrimidine-3-carbonitrile, FE (III) ION, ... (4 entities in total)
Functional Keywordskdm4d, inhibitor, complex, oxidoreductase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight38374.21
Authors
Wang, T.,Yang, L. (deposition date: 2021-01-22, release date: 2022-01-26, Last modification date: 2023-11-29)
Primary citationWang, T.,Yang, L.
Crystal structure of histone lysine demethylase 4D (KDM4D) in complex with the inhibitor 5-hydroxy-2-methylpyrazolo[1,5-a]pyrido[3,2-e]pyrimidine-3-carbonitrile
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.998 Å)
Structure validation

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