7BL9
BAZ2A bromodomain in complex with GSK2801 chemical probe
Summary for 7BL9
Entry DOI | 10.2210/pdb7bl9/pdb |
Related | 4RVR 7BL8 |
Descriptor | Bromodomain adjacent to zinc finger domain protein 2A, 1-{1-[2-(methylsulfonyl)phenyl]-7-propoxyindolizin-3-yl}ethanone, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | four helical bundle, transcription |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 12814.44 |
Authors | Dalle Vedove, A.,Cazzanelli, G.,Caflisch, A.,Lolli, G. (deposition date: 2021-01-18, release date: 2022-03-02, Last modification date: 2024-01-31) |
Primary citation | Cazzanelli, G.,Dalle Vedove, A.,D'Agostino, V.G.,Caflisch, A.,Lolli, G. Chemical probes in the BAZ2A bromodomain to be published, |
Experimental method | X-RAY DIFFRACTION (1.3 Å) |
Structure validation
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