7BL9
BAZ2A bromodomain in complex with GSK2801 chemical probe
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 16 |
Details | binding site for residue 3WQ A 1901 |
Chain | Residue |
A | TRP1816 |
A | LEU1863 |
A | ASP1867 |
A | ASN1873 |
A | VAL1879 |
A | TRP1894 |
A | HOH2014 |
A | HOH2056 |
A | PRO1817 |
A | PHE1818 |
A | GLU1820 |
A | PRO1821 |
A | VAL1822 |
A | VAL1827 |
A | ALA1859 |
A | ALA1860 |
site_id | AC2 |
Number of Residues | 5 |
Details | binding site for residue EDO A 1902 |
Chain | Residue |
A | ARG1846 |
A | ASP1861 |
A | LEU1864 |
A | GLU1878 |
A | HOH2021 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 58 |
Details | BROMODOMAIN_1 Bromodomain signature. AwpFlepvNprlvs..GYRriIknpMdfstMrerllrgg..Ytsseefaadall.VfdNCqtF |
Chain | Residue | Details |
A | ALA1815-PHE1872 |