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7BFZ

X-ray structure of human prostate-specific membrane antigen(PSMA) in complex with a inhibitor Glu-490

Summary for 7BFZ
Entry DOI10.2210/pdb7bfz/pdb
DescriptorGlutamate carboxypeptidase 2, 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, ... (14 entities in total)
Functional Keywordsglutamate carboxypeptidase ii (gcpii); naaladase; prostate-specific membrane antigen (psma); inhibitor, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight84540.56
Authors
Rakhimbekova, A.,Motlova, L.,Barinka, C. (deposition date: 2021-01-05, release date: 2021-08-18, Last modification date: 2024-01-31)
Primary citationZhang, J.,Rakhimbekova, A.,Duan, X.,Yin, Q.,Foss, C.A.,Fan, Y.,Xu, Y.,Li, X.,Cai, X.,Kutil, Z.,Wang, P.,Yang, Z.,Zhang, N.,Pomper, M.G.,Wang, Y.,Barinka, C.,Yang, X.
A prostate-specific membrane antigen activated molecular rotor for real-time fluorescence imaging.
Nat Commun, 12:5460-5460, 2021
Cited by
PubMed: 34526506
DOI: 10.1038/s41467-021-25746-6
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.73 Å)
Structure validation

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