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7ATS

The LIMK1 Kinase Domain Bound To LIJTF500127

Summary for 7ATS
Entry DOI10.2210/pdb7ats/pdb
DescriptorLIM domain kinase 1, N-[3-[5-(4-Chlorophenyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]benzenesulfonamide (2 entities in total)
Functional Keywordskinase inhibitor active site cfl1 actin cytoskeleton, signaling protein
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight36518.71
Authors
Mathea, S.,Chatterjee, D.,Preuss, F.,Yamamoto, S.,Tawada, M.,Nomura, I.,Takagi, T.,Ahmed, M.,Little, W.,Mueller-Knapp, S.,Knapp, S. (deposition date: 2020-10-30, release date: 2020-11-25, Last modification date: 2024-01-31)
Primary citationMathea, S.,Chatterjee, D.,Preuss, F.,Yamamoto, S.,Tawada, M.,Nomura, I.,Takagi, T.,Ahmed, M.,Little, W.,Mueller-Knapp, S.,Knapp, S.
The LIMK1 Kinase Domain Bound To LIJTF500127
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.8 Å)
Structure validation

221051

数据于2024-06-12公开中

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