7Q2M
Crystal structure of the C-terminal catalytic domain of Plasmodium falciparum CTP:phosphocholine cytidylyltransferase with but-3-yn-2-amine hydrochloride
Summary for 7Q2M
Entry DOI | 10.2210/pdb7q2m/pdb |
Descriptor | Cholinephosphate cytidylyltransferase, (2S)-but-3-yn-2-amine (3 entities in total) |
Functional Keywords | plasmodium falciparum cct inhibitors fragments, transferase |
Biological source | Plasmodium falciparum (malaria parasite P. falciparum) |
Total number of polymer chains | 1 |
Total formula weight | 20948.33 |
Authors | Duclovel, C.,Gelin, M.,Krimm, I.,Cerdan, R.,Guichou, J.F. (deposition date: 2021-10-25, release date: 2022-11-23, Last modification date: 2024-01-31) |
Primary citation | Duclovel, C.,Gelin, M.,Wein, S.,Wengelnik, K.,Krimm, I.,Guichou, J.F.,Cerdan, R. Crystallographic screening using ultra-low-molecular-weight ligands to guide drug design of PfCCT inhibitors. To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.08 Å) |
Structure validation
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