7OPG
Crystal structure of CLK1 in complex with compound 2 (CC513)
Summary for 7OPG
Entry DOI | 10.2210/pdb7opg/pdb |
Descriptor | Dual specificity protein kinase CLK1, 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol, GLYCEROL, ... (6 entities in total) |
Functional Keywords | kinase inhibitor, clk1, splicing kinase, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 3 |
Total formula weight | 120916.75 |
Authors | Chaikuad, A.,Routier, S.,Bonnet, P.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2021-05-31, release date: 2021-07-21, Last modification date: 2024-01-31) |
Primary citation | Chaikuad, A.,Routier, S.,Bonnet, P.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of CLK1 in complex with compound 2 (CC513) To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.93 Å) |
Structure validation
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