7LRY
Structure of HIV-1 Reverse Transcriptase in complex with DNA, (-)FTC-TP, and CA(2+) ion
Summary for 7LRY
Entry DOI | 10.2210/pdb7lry/pdb |
Descriptor | Reverse transcriptase p66, [[(2R,5S)-5-(4-azanyl-5-fluoranyl-2-oxidanylidene-pyrimidin-1-yl)-1,3-oxathiolan-2-yl]methoxy-oxidanyl-phosphoryl] phosphono hydrogen phosphate, Reverse transcriptase p51, ... (11 entities in total) |
Functional Keywords | human immunodeficiency virus 1, protein/dsdna, aptamer, dntp, transferase, transferase-dna complex, transferase/dna |
Biological source | Human immunodeficiency virus type 1 (HIV-1) More |
Total number of polymer chains | 6 |
Total formula weight | 254833.14 |
Authors | Hoang, A.,Ruiz, F.X.,Arnold, E. (deposition date: 2021-02-17, release date: 2022-02-23, Last modification date: 2023-10-18) |
Primary citation | Ruiz, F.X.,Hoang, A.,Dilmore, C.R.,DeStefano, J.J.,Arnold, E. Structural basis of HIV inhibition by L-nucleosides: Opportunities for drug development and repurposing. Drug Discov Today, 27:1832-1846, 2022 Cited by PubMed: 35218925DOI: 10.1016/j.drudis.2022.02.016 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.45 Å) |
Structure validation
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