7F8Y
Crystal structure of the cholecystokinin receptor CCKAR in complex with devazepide
Summary for 7F8Y
Entry DOI | 10.2210/pdb7f8y/pdb |
Descriptor | fusion protein of Cholecystokinin receptor type A and Endolysin, N-[(3S)-1-methyl-2-oxidanylidene-5-phenyl-3H-1,4-benzodiazepin-3-yl]-1H-indole-2-carboxamide (2 entities in total) |
Functional Keywords | g protein-coulped receptor, cholecystokinin receptor cckar, devazepide, structural protein |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 1 |
Total formula weight | 60858.82 |
Authors | |
Primary citation | Zhang, X.,He, C.,Wang, M.,Zhou, Q.,Yang, D.,Zhu, Y.,Feng, W.,Zhang, H.,Dai, A.,Chu, X.,Wang, J.,Yang, Z.,Jiang, Y.,Sensfuss, U.,Tan, Q.,Han, S.,Reedtz-Runge, S.,Xu, H.E.,Zhao, S.,Wang, M.W.,Wu, B.,Zhao, Q. Structures of the human cholecystokinin receptors bound to agonists and antagonists. Nat.Chem.Biol., 17:1230-1237, 2021 Cited by PubMed: 34556863DOI: 10.1038/s41589-021-00866-8 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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