7F5E
Crystal structure of BPTF-BRD with ligand DC-BPi-11 bound
Summary for 7F5E
Entry DOI | 10.2210/pdb7f5e/pdb |
Descriptor | Nucleosome-remodeling factor subunit BPTF, N,N-dimethyl-3-[5-(2-methylsulfonyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)indol-1-yl]propan-1-amine (3 entities in total) |
Functional Keywords | bptf bromodomain, lysine acetylation, small-molecule inhibitor, biosynthetic protein, antitumor protein |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 13783.78 |
Authors | |
Primary citation | Lu, T.,Lu, H.B.,Wang, J.,Han, J.,Xiao, S.,Jiang, H.,Chen, Y.,Yang, F.,Li, Q.,Jiang, H.L.,Chen, K.X.,Lu, W.C.,Lin, H.,Luo, C. Discovery and Optimization of Small-Molecule Inhibitors for the BPTF Bromodomains Proteins To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.20017124371 Å) |
Structure validation
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