7AMH
SmBRD3(2), Second Bromodomain of Bromodomain 3 from Schistosoma mansoni in complex with DM-A-33, an iBET726 analogue
Summary for 7AMH
Entry DOI | 10.2210/pdb7amh/pdb |
Descriptor | Putative bromodomain-containing protein 3, brd3, 4-{(2S, 4R)-1-acetyl-4-[(1-benzothiophen-6-yl)amino]-2-methyl-1,2,3,4-tetrahydroquinolin-6-yl}benzoic acid (3 entities in total) |
Functional Keywords | bromo domain, methyllysine binding, epigenetic reader domain, inhibitor, complex, protein binding |
Biological source | Schistosoma mansoni (Blood fluke) |
Total number of polymer chains | 2 |
Total formula weight | 30972.97 |
Authors | McArdle, D.,Schiedel, M.,McDonough, M.A.,Conway, S.J. (deposition date: 2020-10-08, release date: 2021-10-20, Last modification date: 2024-01-31) |
Primary citation | McArdle, D.J.B.,Schiedel, M.,McDonough, M.A.,Conway, S.J. SBM3_2, Second Bromodomain of Bromodomain 3 from Schistosoma mansoni in complex with DM1, an iBET726 analogue To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.863 Å) |
Structure validation
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