6ZFS
Crystal structure of bovine cytochrome bc1 in complex with quinolone inhibitor WDH-1U-4
Summary for 6ZFS
Entry DOI | 10.2210/pdb6zfs/pdb |
Descriptor | Cytochrome b-c1 complex subunit 1, mitochondrial, Cytochrome b-c1 complex subunit 9, 1,2-DIHEXANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, ... (22 entities in total) |
Functional Keywords | cytochrome bc1, malaria, electron transport |
Biological source | Bos taurus (cattle) More |
Total number of polymer chains | 10 |
Total formula weight | 239155.26 |
Authors | Amporndanai, K.,O'Neill, P.M.,Hong, W.D.,Amewu, R.K.,Pidathala, C.,Berry, N.G.,Biagini, G.A.,Leung, S.C.,Hasnain, S.S.,Antonyuk, S.V. (deposition date: 2020-06-17, release date: 2021-06-30, Last modification date: 2024-01-24) |
Primary citation | Amporndanai, K.,O'Neill, P.M.,Hong, W.D.,Amewu, R.K.,Pidathala, C.,Berry, N.,Biangini, G.A.,Leung, S.C.,Hasnain, S.S.,Antonyuk, S.V. Targeting the ubiquinol-reduction (Qi) site of the mitochondrial cytochrome bc1 complex for the development of next generation quinolone antimalarials To Be Published, |
Experimental method | X-RAY DIFFRACTION (3.5 Å) |
Structure validation
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