6ZEL
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound F5
This is a non-PDB format compatible entry.
Summary for 6ZEL
Entry DOI | 10.2210/pdb6zel/pdb |
Descriptor | Bromodomain-containing protein 4, 1,2-ETHANEDIOL, 3,5-dimethyl-4-[(6-methylpyrimidin-4-yl)sulfanylmethyl]-1,2-oxazole, ... (4 entities in total) |
Functional Keywords | bromodomain-containing protein 4 isoform long, brd4, bromodomain-containing protein 4, cap, hunk1, mcap, mitotic chromosome associated protein, cell cycle |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 15520.89 |
Authors | Krojer, T.,Martinez-Cartro, M.,Picaud, S.,Filippakopoulos, P.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Barril, X.,von Delft, F. (deposition date: 2020-06-16, release date: 2020-07-29, Last modification date: 2024-01-24) |
Primary citation | Martinez-Cartro, M.,Barril, X. CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound F5 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.12 Å) |
Structure validation
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