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6ZEL

CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound F5

This is a non-PDB format compatible entry.
Summary for 6ZEL
Entry DOI10.2210/pdb6zel/pdb
DescriptorBromodomain-containing protein 4, 1,2-ETHANEDIOL, 3,5-dimethyl-4-[(6-methylpyrimidin-4-yl)sulfanylmethyl]-1,2-oxazole, ... (4 entities in total)
Functional Keywordsbromodomain-containing protein 4 isoform long, brd4, bromodomain-containing protein 4, cap, hunk1, mcap, mitotic chromosome associated protein, cell cycle
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15520.89
Authors
Krojer, T.,Martinez-Cartro, M.,Picaud, S.,Filippakopoulos, P.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Barril, X.,von Delft, F. (deposition date: 2020-06-16, release date: 2020-07-29, Last modification date: 2024-01-24)
Primary citationMartinez-Cartro, M.,Barril, X.
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound F5
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.12 Å)
Structure validation

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