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6ZCR

SYK Kinase domain in complex with azabenzimidazole inhibitor 7

Summary for 6ZCR
Entry DOI10.2210/pdb6zcr/pdb
DescriptorTyrosine-protein kinase SYK, 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-N-(piperidin-4-ylmethyl)-3H-imidazo[4,5-b]pyridin-7-amine (3 entities in total)
Functional Keywordssyk kinase transferase inhibitor, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight35300.85
Authors
Read, J.A.,Patel, J. (deposition date: 2020-06-12, release date: 2021-06-23, Last modification date: 2024-01-24)
Primary citationRead, J.A.
SYK Kinase domain in complex with azabenzimidazole inhibitor 7
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.73 Å)
Structure validation

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