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6ZCQ

SYK Kinase domain in complex with diamine inhibitor 5

Summary for 6ZCQ
Entry DOI10.2210/pdb6zcq/pdb
DescriptorTyrosine-protein kinase SYK, 7-[[4-[4-[[(3~{R},4~{R})-3-azanyloxan-4-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]-~{N},3-dimethyl-imidazo[1,5-a]pyridine-1-carboxamide (3 entities in total)
Functional Keywordssyk kinase transferase inhibitor, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight35343.48
Authors
Read, J.A. (deposition date: 2020-06-11, release date: 2021-06-23, Last modification date: 2024-01-24)
Primary citationRead, J.A.
SYK Kinase domain in complex with diamine inhibitor 5
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.32 Å)
Structure validation

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