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6Z4M

A4V mutant of human SOD1 bound with 2-(pyridin-3-ylmethyl)benzoisoselenazolone derivative 10 in P21 space group

This is a non-PDB format compatible entry.
Summary for 6Z4M
Entry DOI10.2210/pdb6z4m/pdb
DescriptorSuperoxide dismutase [Cu-Zn], ~{N}-[(6-methoxypyridin-3-yl)methyl]-2-selanyl-benzamide, ZINC ION, ... (6 entities in total)
Functional Keywordssod1, ebselen, motor neuron disease, oxidoreductase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight32782.30
Authors
Amporndanai, K.,Hasnain, S.S. (deposition date: 2020-05-25, release date: 2020-09-16, Last modification date: 2024-01-24)
Primary citationAmporndanai, K.,Rogers, M.,Watanabe, S.,Yamanaka, K.,O'Neill, P.M.,Hasnain, S.S.
Novel Selenium-based compounds with therapeutic potential for SOD1-linked amyotrophic lateral sclerosis.
Ebiomedicine, 59:102980-102980, 2020
Cited by
PubMed: 32862101
DOI: 10.1016/j.ebiom.2020.102980
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.55 Å)
Structure validation

217705

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