6YSY
Skeletal Myosin bound to MPH-220, MgADP-VO4
Summary for 6YSY
Entry DOI | 10.2210/pdb6ysy/pdb |
Descriptor | Myosin-4, Myosin light chain 1/3, skeletal muscle isoform, ADENOSINE-5'-DIPHOSPHATE, ... (7 entities in total) |
Functional Keywords | myofibril, muscle spasticity, actin binding, inhibitor, motor protein |
Biological source | Oryctolagus cuniculus (Rabbit) More |
Total number of polymer chains | 2 |
Total formula weight | 245409.77 |
Authors | Canon, L.,Kikuti, C.M.,Gyimesi, M.,Malnasi-Csizmadia, A.,Houdusse, A. (deposition date: 2020-04-23, release date: 2021-03-03, Last modification date: 2024-01-24) |
Primary citation | Gyimesi, M.,Horvath, A.I.,Turos, D.,Suthar, S.K.,Penzes, M.,Kurdi, C.,Canon, L.,Kikuti, C.,Ruppel, K.M.,Trivedi, D.V.,Spudich, J.A.,Lorincz, I.,Rauscher, A.A.,Kovacs, M.,Pal, E.,Komoly, S.,Houdusse, A.,Malnasi-Csizmadia, A. Single Residue Variation in Skeletal Muscle Myosin Enables Direct and Selective Drug Targeting for Spasticity and Muscle Stiffness. Cell, 183:335-346.e13, 2020 Cited by PubMed: 33035452DOI: 10.1016/j.cell.2020.08.050 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.246 Å) |
Structure validation
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