6YGS
tRNA-guanine Transglycosylase (TGT) in co-crystallized complex with 6-amino-2-(methylamino)-4-(4-(trifluoromethyl)phenethyl)-3,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one
Summary for 6YGS
Entry DOI | 10.2210/pdb6ygs/pdb |
Related | 6YGR |
Descriptor | Queuine tRNA-ribosyltransferase, ZINC ION, 6-amino-2-(methylamino)-4-(4-(trifluoromethyl)phenethyl)-3,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one, ... (5 entities in total) |
Functional Keywords | transferase, tgt, trna-guanine transglycosylase, guanine insertion enzyme, homodimer |
Biological source | Zymomonas mobilis subsp. mobilis (strain ATCC 31821 / ZM4 / CP4) |
Total number of polymer chains | 1 |
Total formula weight | 43629.70 |
Authors | Nguyen, A.,Heine, A.,Klebe, G. (deposition date: 2020-03-27, release date: 2020-04-08, Last modification date: 2024-01-24) |
Primary citation | Nguyen, A.,Heine, A.,Klebe, G. Co-crystallization and 19F NMR reveal dimer disturbing inhibitors and conformational changes at dimer contacts To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.4 Å) |
Structure validation
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