6XER
Tubulin-RB3_SLD in complex with colchicine
Summary for 6XER
Entry DOI | 10.2210/pdb6xer/pdb |
Descriptor | Tubulin alpha-1B chain, Tubulin beta chain, Stathmin-4, ... (9 entities in total) |
Functional Keywords | microtubule inhibitor, colchicine, cell cycle, cancer, cell cycle-inhibitor complex, cell cycle/inhibitor |
Biological source | Rattus norvegicus (Rat) More |
Total number of polymer chains | 5 |
Total formula weight | 214857.09 |
Authors | White, S.W.,Yun, M. (deposition date: 2020-06-13, release date: 2021-08-25, Last modification date: 2023-10-18) |
Primary citation | Chen, H.,Deng, S.,Albadari, N.,Yun, M.K.,Zhang, S.,Li, Y.,Ma, D.,Parke, D.N.,Yang, L.,Seagroves, T.N.,White, S.W.,Miller, D.D.,Li, W. Design, Synthesis, and Biological Evaluation of Stable Colchicine-Binding Site Tubulin Inhibitors 6-Aryl-2-benzoyl-pyridines as Potential Anticancer Agents. J.Med.Chem., 64:12049-12074, 2021 Cited by PubMed: 34378386DOI: 10.1021/acs.jmedchem.1c00715 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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