6WV5
Human VKOR C43S mutant with vitamin K1 epoxide
Summary for 6WV5
Entry DOI | 10.2210/pdb6wv5/pdb |
Descriptor | Vitamin K epoxide reductase Cys43Ser mutant, termini restrained by green fluorescent protein, (2R,3R)-2-hydroxy-3-methyl-2-[(2E,7S)-3,7,11,15-tetramethylhexadec-2-en-1-yl]-2,3-dihydronaphthalene-1,4-dione (2 entities in total) |
Functional Keywords | vitamin k epoxide reductase (vkor), vitamin k, warfarin, superwarfarin, vitamin k expoxide(ko), membrane protein, oxidoreductase, fluorescent protein |
Biological source | Aequorea victoria (Jellyfish) More |
Total number of polymer chains | 1 |
Total formula weight | 44650.08 |
Authors | Liu, S.,Sukumar, N.,Li, W. (deposition date: 2020-05-05, release date: 2020-11-11, Last modification date: 2023-11-15) |
Primary citation | Liu, S.,Li, S.,Shen, G.,Sukumar, N.,Krezel, A.M.,Li, W. Structural basis of antagonizing the vitamin K catalytic cycle for anticoagulation. Science, 371:-, 2021 Cited by PubMed: 33154105DOI: 10.1126/science.abc5667 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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