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6V87

Estrogen Receptor Alpha Ligand Binding Domain Y537S in Complex with 4-Hydroxytamoxifen

Summary for 6V87
Entry DOI10.2210/pdb6v87/pdb
DescriptorEstrogen receptor, 4-HYDROXYTAMOXIFEN (3 entities in total)
Functional Keywordsestrogen receptor, serm, activating mutation, breast cancer, transcription
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight60843.09
Authors
Fanning, S.W.,Greene, G.L. (deposition date: 2019-12-10, release date: 2019-12-25, Last modification date: 2023-10-11)
Primary citationFanning, S.W.
Estrogen Receptor Alpha
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

222624

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