6V87
Estrogen Receptor Alpha Ligand Binding Domain Y537S in Complex with 4-Hydroxytamoxifen
Summary for 6V87
Entry DOI | 10.2210/pdb6v87/pdb |
Descriptor | Estrogen receptor, 4-HYDROXYTAMOXIFEN (3 entities in total) |
Functional Keywords | estrogen receptor, serm, activating mutation, breast cancer, transcription |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 60843.09 |
Authors | Fanning, S.W.,Greene, G.L. (deposition date: 2019-12-10, release date: 2019-12-25, Last modification date: 2023-10-11) |
Primary citation | Fanning, S.W. Estrogen Receptor Alpha To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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