6UL9
Crystal structure of human GAC in complex with inhibitor UPGL00023
Summary for 6UL9
Entry DOI | 10.2210/pdb6ul9/pdb |
Descriptor | Glutaminase kidney isoform, mitochondrial, 2-phenyl-N-{5-[(1-{5-[(phenylacetyl)amino]-1,3,4-thiadiazol-2-yl}azetidin-3-yl)oxy]-1,3,4-thiadiazol-2-yl}acetamide (3 entities in total) |
Functional Keywords | inhibitor, complex, hydrolase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 4 |
Total formula weight | 233223.35 |
Authors | Huang, Q.Q.,Cerione, R.A. (deposition date: 2019-10-07, release date: 2020-10-14, Last modification date: 2023-10-11) |
Primary citation | Huang, Q.,Cerione, R.A. Crystal structure of human GAC in complex with inhibitor UPGL00012 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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