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6UIM

Crystal Structure of Danio rerio Histone Deacetylase 10 in Complex with 7-{[(3-aminopropyl)amino]-2-oxoheptyl} thioacetate

Summary for 6UIM
Entry DOI10.2210/pdb6uim/pdb
DescriptorPolyamine deacetylase HDAC10, 7-[(3-aminopropyl)amino]-1-sulfanylheptan-2-one, ZINC ION, ... (6 entities in total)
Functional Keywordshistone deacetylase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceDanio rerio
Total number of polymer chains1
Total formula weight75593.51
Authors
Herbst-Gervasoni, C.J.,Christianson, D.W. (deposition date: 2019-10-01, release date: 2019-12-04, Last modification date: 2023-10-11)
Primary citationHerbst-Gervasoni, C.J.,Christianson, D.W.
Binding ofN8-Acetylspermidine Analogues to Histone Deacetylase 10 Reveals Molecular Strategies for Blocking Polyamine Deacetylation.
Biochemistry, 58:4957-4969, 2019
Cited by
PubMed: 31746596
DOI: 10.1021/acs.biochem.9b00906
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.75 Å)
Structure validation

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