6TX4
CRYSTAL STRUCTURE OF HUMAN FKBP51 FK1 DOMAIN A19T MUTANT IN COMPLEX WITH 2-PYRIDONE
Summary for 6TX4
Entry DOI | 10.2210/pdb6tx4/pdb |
Descriptor | Peptidyl-prolyl cis-trans isomerase FKBP5, CHLORIDE ION, SODIUM ION, ... (5 entities in total) |
Functional Keywords | ppiase, fragment, isomerase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 14297.71 |
Authors | Fiegen, D.,Draxler, S.W. (deposition date: 2020-01-13, release date: 2020-05-27, Last modification date: 2024-01-24) |
Primary citation | Draxler, S.W.,Bauer, M.,Eickmeier, C.,Nadal, S.,Nar, H.,Rangel Rojas, D.,Seeliger, D.,Zeeb, M.,Fiegen, D. Hybrid Screening Approach for Very Small Fragments: X-ray and Computational Screening on FKBP51. J.Med.Chem., 63:5856-5864, 2020 Cited by PubMed: 32420743DOI: 10.1021/acs.jmedchem.0c00120 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.06 Å) |
Structure validation
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