6TW8

Leishmania major N-myristoyltransferase in complex with indazole inhibitor IMP-917

This is a non-PDB format compatible entry.

Summary for 6TW8

• Entry DOI: 10.2210/pdb6tw8/pdb
• Related: 5O6H
• Descriptor: Glycylpeptide N-tetradecanoyltransferase, TETRADECANOYL-COA, 1-[5-[4-fluoranyl-2-[2-(1,3,5-trimethylpyrazol-4-yl)ethoxy]phenyl]-2~{H}-indazol-3-yl]-~{N},~{N}-dimethyl-methanamine, ... (5 entities in total)
• Functional Keywords: transferase, myristoylation, indazole, leishmania
• Biological source: Leishmania major
• Total number of polymer chains: 2
• Total formula weight: 99238.95

Authors

Brannigan, J.A. (deposition date: 2020-01-12, release date: 2021-07-21, Last modification date: 2024-05-15)

• Primary citation: Brannigan, J.A.; Leishmania major N-myristoyltransferase in complex with indazole inhibitor IMP-917; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.79 Å)