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6T1V

Structure of PPARg H494Y mutant in complex with GW1929

Summary for 6T1V
Entry DOI10.2210/pdb6t1v/pdb
DescriptorPeroxisome proliferator-activated receptor gamma, Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, (2~{S})-3-[4-[2-[methyl(pyridin-2-yl)amino]ethoxy]phenyl]-2-[[2-(phenylcarbonyl)phenyl]amino]propanoic acid, ... (4 entities in total)
Functional Keywordsnuclear receptor, complex, transcription
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight33907.44
Authors
Rochel, N. (deposition date: 2019-10-06, release date: 2021-04-14, Last modification date: 2024-02-07)
Primary citationRochel, N.
Structure of a PPARg mutant complex
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.21 Å)
Structure validation

221051

건을2024-06-12부터공개중

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