Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6T1V

Structure of PPARg H494Y mutant in complex with GW1929

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1APeroxisome proliferator-activated receptor gammapolymer27931888.01UniProt (P37231)
Pfam (PF00104)
In PDB
Homo sapiens (human)PPAR-gamma,Nuclear receptor subfamily 1 group C member 3
2CPeroxisome proliferator-activated receptor gamma coactivator 1-alphapolymer141523.91UniProt (Q9UBK2)
In PDB
Homo sapiensPPARGC-1-alpha,Ligand effect modulator 6
3A(2~{S})-3-[4-[2-[methyl(pyridin-2-yl)amino]ethoxy]phenyl]-2-[[2-(phenylcarbonyl)phenyl]amino]propanoic acidnon-polymer495.61Chemie (EDK)
4waterwater18.0230Chemie (HOH)
Sequence modifications
A: 231 - 505 (UniProt: P37231)
PDBExternal DatabaseDetails
Gly 227-expression tag
Ser 228-expression tag
His 229-expression tag
Met 230-expression tag
Tyr 494His 494engineered mutation
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains2
Total formula weight33411.9
Non-Polymers*Number of molecules1
Total formula weight495.6
All*Total formula weight33907.4
*Water molecules are not included.

221051

PDB entries from 2024-06-12

PDB statisticsPDBj update infoContact PDBjnumon