6RCG

Crystal structure of Casein kinase 1 delta (CK1 delta) complexed with SR3029 inhibitor

6RCG の概要

• エントリーDOI: 10.2210/pdb6rcg/pdb
• 分子名称: Casein kinase I isoform delta, 1,2-ETHANEDIOL, ~{N}-[[6,7-bis(fluoranyl)-1~{H}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amine, ... (4 entities in total)
• 機能のキーワード: csnk1d, ck1 delta, ck1d, kinase inhibitor, structural genomics, structural genomics consortium, sgc, transferase
• 由来する生物種: Homo sapiens (Human)
• タンパク質・核酸の鎖数: 1
• 化学式量合計: 35029.39

構造登録者

Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2019-04-11, 公開日: 2020-03-25, 最終更新日: 2024-01-24)

• 主引用文献: Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC); Crystal structure of Casein kinase 1 delta (CK1 delta) complexed with SR3029 inhibitor; To Be Published,

実験手法

X-RAY DIFFRACTION (1.4 Å)