6RAA
CLK1 Kinase domain with bound imidazopyridin inhibitor TP003
Summary for 6RAA
Entry DOI | 10.2210/pdb6raa/pdb |
Descriptor | Dual specificity protein kinase CLK1, 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{N}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | inhibitor, kinase, transferase, structural genomics, structural genomics consortium, sgc |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 40126.16 |
Authors | Schroeder, M.,Arrowsmith, C.,Knapp, S.,Bountra, C.,Edwards, A.,Structural Genomics Consortium (SGC) (deposition date: 2019-04-05, release date: 2019-04-24, Last modification date: 2024-01-24) |
Primary citation | Schroeder, M.,Arrowsmith, C.,Knapp, S.,Bountra, C.,Edwards, A. CLK1 Kinase domain with bound imidazopyridin inhibitor TP003 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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