6QY9
Human CSNK2A2 bound to a Pyrrolo[2,3-d]pyrimidinyl inhibitor
Summary for 6QY9
Entry DOI | 10.2210/pdb6qy9/pdb |
Descriptor | Casein kinase II subunit alpha', 3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrile, 1,2-ETHANEDIOL, ... (5 entities in total) |
Functional Keywords | kinase, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 40495.17 |
Authors | Abdul Azeez, K.R.,Sorrell, F.J.,Krojer, T.,Bountra, C.,Edwards, A.M.,Arrowsmith, C.,Knapp, S.,Elkins, J.M. (deposition date: 2019-03-08, release date: 2019-04-17, Last modification date: 2024-01-24) |
Primary citation | Abdul Azeez, K.R.,Elkins, J.M. Human CSNK2A2 bound to a Pyrrolo[2,3-d]pyrimidinyl inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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