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6QY9

Human CSNK2A2 bound to a Pyrrolo[2,3-d]pyrimidinyl inhibitor

Summary for 6QY9
Entry DOI10.2210/pdb6qy9/pdb
DescriptorCasein kinase II subunit alpha', 3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrile, 1,2-ETHANEDIOL, ... (5 entities in total)
Functional Keywordskinase, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight40495.17
Authors
Abdul Azeez, K.R.,Sorrell, F.J.,Krojer, T.,Bountra, C.,Edwards, A.M.,Arrowsmith, C.,Knapp, S.,Elkins, J.M. (deposition date: 2019-03-08, release date: 2019-04-17, Last modification date: 2024-01-24)
Primary citationAbdul Azeez, K.R.,Elkins, J.M.
Human CSNK2A2 bound to a Pyrrolo[2,3-d]pyrimidinyl inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

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