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6QJ7

Difluorophenyl diacylhydrazides: Potent inhibitors of Serum- and Glucocorticoid-inducible Kinase 1 (SGK1)

Summary for 6QJ7
Entry DOI10.2210/pdb6qj7/pdb
Related2GU8
DescriptorcAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha, ~{N}'-[(2~{S})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazide, ... (4 entities in total)
Functional Keywordscamp-dependent protein kinase a (pka), transferase
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight43399.32
Authors
Graedler, U. (deposition date: 2019-01-23, release date: 2020-02-12, Last modification date: 2024-11-20)
Primary citationGraedler, U.
Difluorophenyl diacylhydrazides: Potent inhibitors of Serum- and Glucocorticoid-inducible Kinase 1 (SGK1)
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.69 Å)
Structure validation

227561

PDB entries from 2024-11-20

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