6QE1
P38 alpha complex with AR117046
Summary for 6QE1
Entry DOI | 10.2210/pdb6qe1/pdb |
Related | 6QDZ |
Descriptor | Mitogen-activated protein kinase 14, 2-fluoro-4-[4-(4-fluorophenyl)-1H-pyrazol-3-yl]pyridine, 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{S},4~{R})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea, ... (4 entities in total) |
Functional Keywords | inhibitor, complex, kinase, signaling protein |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 42322.28 |
Authors | Brown, D.G.,Hurley, C.,Irving, S.L. (deposition date: 2019-01-03, release date: 2020-01-29, Last modification date: 2024-05-15) |
Primary citation | Brown, D.G.,Irving, S.L. P38 alpha complex with AR117045 and AR117046 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.85 Å) |
Structure validation
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