6Q55
Crystal structure of Cryptosporidium hominis CPSF3 in complex with Compound 61
Summary for 6Q55
Entry DOI | 10.2210/pdb6q55/pdb |
Descriptor | Cleavage and Polyadenylation Specificity Factor 3 (CPSF3), ZINC ION, 3-[7,7-bis(oxidanyl)-8-oxa-7-boranuidabicyclo[4.3.0]nona-1(6),2,4-trien-5-yl]propanoic acid, ... (7 entities in total) |
Functional Keywords | mrna processing factor, metallo-beta-lactamase, beta-casp, oxaborole-inhibitor, rna binding protein |
Biological source | Cryptosporidium hominis TU502 |
Total number of polymer chains | 1 |
Total formula weight | 55113.32 |
Authors | Palencia, A.,Swale, C. (deposition date: 2018-12-07, release date: 2019-11-20, Last modification date: 2024-01-24) |
Primary citation | Swale, C.,Bougdour, A.,Gnahoui-David, A.,Tottey, J.,Georgeault, S.,Laurent, F.,Palencia, A.,Hakimi, M.A. Metal-captured inhibition of pre-mRNA processing activity by CPSF3 controls Cryptosporidium infection. Sci Transl Med, 11:-, 2019 Cited by PubMed: 31694928DOI: 10.1126/scitranslmed.aax7161 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
Download full validation report