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6Q2A

Trypanosoma brucei CLK1 kinase domain in complex with a covalent aminobenzimidazole inhibitor AB1

Summary for 6Q2A
Entry DOI10.2210/pdb6q2a/pdb
DescriptorProtein kinase, putative, SULFATE ION, ~{N}-[1-[(3~{R})-1-[4-(dimethylamino)but-2-enoyl]azepan-3-yl]-7-methyl-benzimidazol-2-yl]-2-methyl-pyridine-4-carboxamide, ... (4 entities in total)
Functional Keywordskinase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceTrypanosoma brucei brucei (strain 927/4 GUTat10.1)
Total number of polymer chains16
Total formula weight668678.53
Authors
Ma, X.,Ornelas, E. (deposition date: 2019-08-07, release date: 2020-06-17, Last modification date: 2023-10-11)
Primary citationSaldivia, M.,Fang, E.,Ma, X.,Myburgh, E.,Carnielli, J.B.T.,Bower-Lepts, C.,Brown, E.,Ritchie, R.,Lakshminarayana, S.B.,Chen, Y.L.,Patra, D.,Ornelas, E.,Koh, H.X.Y.,Williams, S.L.,Supek, F.,Paape, D.,McCulloch, R.,Kaiser, M.,Barrett, M.P.,Jiricek, J.,Diagana, T.T.,Mottram, J.C.,Rao, S.P.S.
Targeting the trypanosome kinetochore with CLK1 protein kinase inhibitors.
Nat Microbiol, 5:1207-1216, 2020
Cited by
PubMed: 32661312
DOI: 10.1038/s41564-020-0745-6
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.6 Å)
Structure validation

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