6PDN
Human PIM1 bound to benzothiophene inhibitor 292
Summary for 6PDN
Entry DOI | 10.2210/pdb6pdn/pdb |
Related | 6PCW 6PDI |
Descriptor | Serine/threonine-protein kinase pim-1, peptide, 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid, ... (5 entities in total) |
Functional Keywords | proto-oncogene serine/threonine-protein kinase pim-1, structural genomics, structural genomics consortium, sgc, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 37715.87 |
Authors | Godoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M.,Structural Genomics Consortium (SGC) (deposition date: 2019-06-19, release date: 2019-07-24, Last modification date: 2020-01-01) |
Primary citation | Godoi, P.H.C.,Santiago, A.S.,Fala, A.M.,Ramos, P.Z.,Sriranganadane, D.,Mascarello, A.,Segretti, N.,Azevedo, H.,Guimaraes, C.R.W.,Arruda, P.,Elkins, J.M.,Counago, R.M. Human PIM1 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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