6NFT
Structure of USP5 zinc-finger ubiquitin binding domain co-crystallized with (4-oxoquinazolin-3(4H)-yl)acetic acid
Summary for 6NFT
Entry DOI | 10.2210/pdb6nft/pdb |
Related | 6DXH 6DXT |
Descriptor | Ubiquitin carboxyl-terminal hydrolase 5, ZINC ION, (4-oxoquinazolin-3(4H)-yl)acetic acid, ... (6 entities in total) |
Functional Keywords | usp5, structural genomics, structural genomics consortium, sgc, hydrolase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 27795.78 |
Authors | Harding, R.J.,Mann, M.K.,Tempel, W.,Bountra, C.,Arrowmsmith, C.M.,Edwards, A.M.,Schapira, M.,Structural Genomics Consortium (SGC) (deposition date: 2018-12-20, release date: 2019-01-02, Last modification date: 2021-06-09) |
Primary citation | Mann, M.K.,Franzoni, I.,de Freitas, R.F.,Tempel, W.,Houliston, S.,Smith, L.,Vedadi, M.,Arrowsmith, C.H.,Harding, R.J.,Schapira, M. Discovery of Small Molecule Antagonists of the USP5 Zinc Finger Ubiquitin-Binding Domain. J.Med.Chem., 62:10144-10155, 2019 Cited by PubMed: 31663737DOI: 10.1021/acs.jmedchem.9b00988 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.65 Å) |
Structure validation
Download full validation report