6N8G
IRAK4 bound to benzoxazole compound
Summary for 6N8G
| Entry DOI | 10.2210/pdb6n8g/pdb |
| Descriptor | Interleukin-1 receptor-associated kinase 4, N-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1H-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide (3 entities in total) |
| Functional Keywords | protein kinase, irak4, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
| Biological source | Homo sapiens (Human) |
| Total number of polymer chains | 4 |
| Total formula weight | 136309.53 |
| Authors | Larsen, N.A.,Bloudoff, K.,Subramanian, V.,Dobrzanska, M.,Gluza, K. (deposition date: 2018-11-29, release date: 2018-12-12, Last modification date: 2024-10-23) |
| Primary citation | Larsen, N.A.,Gluza, K. To be published To Be Published, |
| Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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