6N87
Plasmodium falciparum FVO apical membrane antigen 1 (AMA1) bound to MTSL spin-labelled cyclised RON2 peptide
Summary for 6N87
Entry DOI | 10.2210/pdb6n87/pdb |
Related | 6N7Q |
Descriptor | Apical membrane antigen-1, backbone-cyclised peptide bcRON2hp, S-[(1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)methyl] methanesulfonothioate, ... (4 entities in total) |
Functional Keywords | ama1, apical membrane antigen 1, malaria, ron2, paramagnetic probe, peptide binding protein |
Biological source | Plasmodium falciparum More |
Total number of polymer chains | 2 |
Total formula weight | 40204.11 |
Authors | McGowan, S.,Drinkwater, N. (deposition date: 2018-11-28, release date: 2019-01-30, Last modification date: 2023-10-11) |
Primary citation | Akter, M.,Drinkwater, N.,Devine, S.M.,Drew, S.C.,Krishnarjuna, B.,Debono, C.O.,Wang, G.,Scanlon, M.J.,Scammells, P.J.,McGowan, S.,MacRaild, C.A.,Norton, R.S. Identification of the Binding Site of Apical Membrane Antigen 1 (AMA1) Inhibitors Using a Paramagnetic Probe. ChemMedChem, 14:603-612, 2019 Cited by PubMed: 30653832DOI: 10.1002/cmdc.201800802 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.588 Å) |
Structure validation
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