6M4W
Crystal structure of MBP fused split FKBP-FRB T2098L mutant in complex with rapamycin
Summary for 6M4W
Entry DOI | 10.2210/pdb6m4w/pdb |
Related PRD ID | PRD_900001 |
Descriptor | chimera of Maltose/maltodextrin-binding periplasmic protein and Peptidyl-prolyl cis-trans isomerase FKBP1A, Peptidyl-prolyl cis-trans isomerase FKBP1A, Serine/threonine-protein kinase mTOR, ... (7 entities in total) |
Functional Keywords | rapamycin, complex, kinase, isomerase |
Biological source | Escherichia coli K-12 More |
Total number of polymer chains | 9 |
Total formula weight | 195887.56 |
Authors | Kikuchi, M.,Wu, D.,Inoue, T.,Umehara, T. (deposition date: 2020-03-09, release date: 2020-08-26, Last modification date: 2023-11-29) |
Primary citation | Wu, H.D.,Kikuchi, M.,Dagliyan, O.,Aragaki, A.K.,Nakamura, H.,Dokholyan, N.V.,Umehara, T.,Inoue, T. Rational design and implementation of a chemically inducible heterotrimerization system. Nat.Methods, 17:928-936, 2020 Cited by PubMed: 32747768DOI: 10.1038/s41592-020-0913-x PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.11 Å) |
Structure validation
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