6LIH

BRD4 BD1 bound with compound 10

Summary for 6LIH

• Entry DOI: 10.2210/pdb6lih/pdb
• Descriptor: Bromodomain-containing protein 4, (3~{R})-1,3-dimethyl-6-[(4-phenylpyrimidin-2-yl)amino]-4-propan-2-yl-3~{H}-quinoxalin-2-one (3 entities in total)
• Functional Keywords: cancer, bromodomain, gene regulation
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 15141.55

Authors

Xiong, B.,Cao, D. (deposition date: 2019-12-11, release date: 2020-12-16, Last modification date: 2023-11-22)

• Primary citation: Xiong, B.,Cao, D.; BRD4 BD1 bound with compound 10; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.6203054097 Å)