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6JYP

Crystal structure of uPA_H99Y in complex with 3-azanyl-5-(azepan-1-yl)-N-[bis(azanyl)methylidene]-6-chloranyl-pyrazine-2-carboxamide

Summary for 6JYP
Entry DOI10.2210/pdb6jyp/pdb
DescriptorUrokinase-type plasminogen activator, 3-azanyl-5-(azepan-1-yl)-N-[bis(azanyl)methylidene]-6-chloranyl-pyrazine-2-carboxamide, SULFATE ION, ... (4 entities in total)
Functional Keywordsurokinase, amiloride, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight28148.46
Authors
Buckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M. (deposition date: 2019-04-27, release date: 2020-05-13, Last modification date: 2024-10-09)
Primary citationBuckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M.
uPA-HMA
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.25 Å)
Structure validation

247947

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