6JTC
Crystal structure of dipeptidyl peptidase 11 (DPP11) with SH-5 from Porphyromonas gingivalis (Space)
Summary for 6JTC
Entry DOI | 10.2210/pdb6jtc/pdb |
Descriptor | Asp/Glu-specific dipeptidyl-peptidase, GLYCEROL, 2-(2-azanylethylamino)-5-nitro-benzoic acid, ... (4 entities in total) |
Functional Keywords | dipeptidyl aminopeptidase, s46, perio, microgravity, antimicrobial, hydrolase |
Biological source | Porphyromonas gingivalis (strain ATCC 33277 / DSM 20709 / CIP 103683 / JCM 12257 / NCTC 11834 / 2561) |
Total number of polymer chains | 2 |
Total formula weight | 164634.90 |
Authors | Sakamoto, Y.,Suzuki, Y.,Iizuka, I.,Roppongi, S.,Kushibiki, C.,Nakamura, A.,Ogasawara, W.,Tanaka, N. (deposition date: 2019-04-10, release date: 2019-10-02, Last modification date: 2023-11-22) |
Primary citation | Sakamoto, Y.,Suzuki, Y.,Nakamura, A.,Watanabe, Y.,Sekiya, M.,Roppongi, S.,Kushibiki, C.,Iizuka, I.,Tani, O.,Sakashita, H.,Inaka, K.,Tanaka, H.,Yamada, M.,Ohta, K.,Honma, N.,Shida, Y.,Ogasawara, W.,Nakanishi-Matsui, M.,Nonaka, T.,Gouda, H.,Tanaka, N. Fragment-based discovery of the first nonpeptidyl inhibitor of an S46 family peptidase. Sci Rep, 9:13587-13587, 2019 Cited by PubMed: 31537874DOI: 10.1038/s41598-019-49984-3 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.39 Å) |
Structure validation
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