6JJ5
BRD4 in complex with 259
Summary for 6JJ5
Entry DOI | 10.2210/pdb6jj5/pdb |
Descriptor | Bromodomain-containing protein 4, 3-((1-methyl-2-oxo-1,2,2a1,5a-tetrahydro-6H-pyrido[3',2':6,7]azepino[4,3,2-cd]isoindol-6-yl)methyl)benzamide (3 entities in total) |
Functional Keywords | brd4, inhibitor, signaling protein-inhibitor complex, signaling protein/inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 15265.60 |
Authors | |
Primary citation | Xu, J.,Zhu, J.,Chen, Y.,Jiang, F. BRD4 in complex with ZZM1 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.2 Å) |
Structure validation
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