6JI4
brd4-bd1 bound with ligand 138
Summary for 6JI4
Entry DOI | 10.2210/pdb6ji4/pdb |
Descriptor | Bromodomain-containing protein 4, (3R)-4-cyclopropyl-1,3-dimethyl-6-[5-methyl-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]-3,4-dihydroquinoxalin-2(1H)-one (3 entities in total) |
Functional Keywords | dna damage, transcription regulation, bromodomain-containing protein 4, transcription |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 15010.36 |
Authors | |
Primary citation | Cao, D.Y.,Li, Y.L.,Du, Z.Y.,Li, J.,Xiong, B. brd4-bd1 bound with ligand 138 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.6 Å) |
Structure validation
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